Search Result "Antimitotic"


Pyridine Based Antitumour Compounds Acting at the Colchicine Site

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 11 Year: 2016 Page: 1100-1130
Author(s): R. Álvarez,L. Aramburu,P. Puebla,E. Caballero,M. González,A. Vicente,M. Medarde,R. Peláez

Synthesis of Chalcone Derivatives and Their Effects on Proliferation and Tubulin Dynamics Instability of HT-29 Cells

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 7 Year: 2016 Page: 662-667
Author(s): Yasmin Tajuddin, Zaliha Harun, Ahmad Rohi Ghazali, Juriyati Jalil, Malina Jasamai

Research Article

Significance of Amino Group Substitution at Combretastatin A-4 and Phenstatin Analogs

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 9 Year: 2016 Page: 943-951
Author(s): Vijay K. Patel, Harish Rajak

Synthesis, Molecular Docking Study, and Cytotoxic Activity of 1,3,5-triaryl Pyrazole Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 2 Year: 2016 Page: 121-128
Author(s): Maryam Ghasemi,Sajad Ghadbeighi,Amirali Amirhamzeh,Seyed AbbasTabatabai,Seyed Nasser Ostad,Abbas Shafiee,Mohsen Amini

A Computational Analysis of Indomethacin Derivative as Tubulin Inhibitor: Insights into Development of Chemotherapeutic Agents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 19 Issue: 6 Year: 2016 Page: 431-436
Author(s): Kelly Miranda Costa,Cláudio Nahum Alves,José Rogério Araújo Silva,Jerônimo Lameira

Review Article

Synthesis of Combretastatin A-4 Analogs and their Biological Activities

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 8 Year: 2016 Page: 942-960
Author(s): Agnieszka Siebert,Monika Gensicka,Grzegorz Cholewinski,Krystyna Dzierzbicka

Metal Containing Cytostatics and Their Interaction with Cellular Thiol Compounds Causing Chemoresistance

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 6 Year: 2016 Page: 686-698
Author(s): Jan Hrabeta,Vojtech Adam,Tomas Eckschlager,Eva Frei,Marie Stiborova,Rene Kizek

1,3,4-oxadiazole-2-thione Derivatives; Novel Approach for Anticancer and Tubulin Polymerization Inhibitory Activities

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 269-277
Author(s): Mohamed Abdel-Aziz,Kamel A. Metwally,Amira M. Gamal-Eldeen,Omar M. Aly

Cyanobacteria as a Source for Novel Anti-Leukemic Compounds

Journal: Current Pharmaceutical Biotechnology
Volume: 17 Issue: 1 Year: 2016 Page: 78-91
Author(s): Anu Humisto,Lars Herfindal,Jouni Jokela,Antti Karkman,Ronja Bjørnstad,Romi R. Choudhury,Kaarina Sivonen

Synthesis, Cytotoxic Evaluation, Docking and QSAR Study of N-(4-Oxo- 2-(4-((5-Aryl-1,3,4-Thiadiazol-2-yl)Amino)Phenyl)Thiazolidin-3-yl) Benzamides as Antitubulin Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 2509-2520
Author(s): Chawla Amit, Chawla Payal, U.S. Baghel, Deep Aakash

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